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Search Results for " histamine h1-receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T7477 Antazoline Others
Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.
T9353 OXOMEMAZINE AChR , Histamine Receptor
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...
T36949 Niaprazine 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff...
T1278 Astemizole Laridal,Histaminos,Paralergin Potassium Channel , Histamine Receptor
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re...
TN1008 Psoralenoside CaMK , Calcium Channel , Histamine Receptor
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.
T0147 Clemastine fumarate HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate) Autophagy , Histamine Receptor
Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T22501 2-Pyridylethylamine dihydrochloride Histamine Receptor
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
T7085 Mebhydrolin Mebhydroline Histamine Receptor
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
T1469 Levocetirizine Levocetirizine HCl Histamine Receptor
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.
T0263 Chloropyramine hydrochloride Nilfan,Alergosan,Halopyramine hydrochloride FAK , VEGFR , Histamine Receptor
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
T23297 (S)-(+)-Dimethindene maleate AChR , Histamine Receptor
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M4 receptors.
T13566 Bamirastine TAK-427 Histamine Receptor
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on allergic skin inflammation.
T22842 HTMT dimaleate Histamine Trifluoromethyl Toluidide Dimaleate Histamine Receptor
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.
T6426 Buclizine dihydrochloride Longifene,Buclina,Buclizine HCl,UCB-4445 5-HT Receptor , AChR , Histamine Receptor
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ...
T1097 Loratadine SCH 29851,Loratidine Influenza Virus , Histamine Receptor
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical antihistamines (HISTAMINE H1 ANTAGONISTS) it lacks central ne...
T22354 Levocetirizine Dihydrochloride Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride Histamine Receptor
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro...
T0092 Antazoline hydrochloride Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl Histamine Receptor
Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous histamine.
T20884 Hydroxyzine Hydroxyzine free base Histamine Receptor
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
T7893 Bepotastine Bepotastine free base Others , Histamine Receptor
Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.
T1115 Doxylamine succinate Decapryn Histamine Receptor
Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties. Doxylamine succinate (Decapryn) competitively blocks the histamine H1 receptor and limits the typical allergic and ...

Compounds

Antazoline
T7477
Synonym:
Target: Others
OXOMEMAZINE
T9353
Synonym:
Target: AChR, Histamine Receptor
Niaprazine
T36949
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Astemizole
T1278
Synonym: Laridal,Histaminos,Paralergin
Target: Potassium Channel, Histamine Receptor
Psoralenoside
TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
Clemastine fumarate
T0147
Synonym: HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate)
Target: Autophagy, Histamine Receptor
2-Pyridylethylamine dihydrochloride
T22501
Synonym:
Target: Histamine Receptor
Mebhydrolin
T7085
Synonym: Mebhydroline
Target: Histamine Receptor
Levocetirizine
T1469
Synonym: Levocetirizine HCl
Target: Histamine Receptor
Chloropyramine hydrochloride
T0263
Synonym: Nilfan,Alergosan,Halopyramine hydrochloride
Target: FAK, VEGFR, Histamine Receptor
(S)-(+)-Dimethindene maleate
T23297
Synonym:
Target: AChR, Histamine Receptor
Bamirastine
T13566
Synonym: TAK-427
Target: Histamine Receptor
HTMT dimaleate
T22842
Synonym: Histamine Trifluoromethyl Toluidide Dimaleate
Target: Histamine Receptor
Buclizine dihydrochloride
T6426
Synonym: Longifene,Buclina,Buclizine HCl,UCB-4445
Target: 5-HT Receptor, AChR, Histamine Receptor
Loratadine
T1097
Synonym: SCH 29851,Loratidine
Target: Influenza Virus, Histamine Receptor
Levocetirizine Dihydrochloride
T22354
Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride
Target: Histamine Receptor
Antazoline hydrochloride
T0092
Synonym: Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl
Target: Histamine Receptor
Hydroxyzine
T20884
Synonym: Hydroxyzine free base
Target: Histamine Receptor
Bepotastine
T7893
Synonym: Bepotastine free base
Target: Others, Histamine Receptor
Doxylamine succinate
T1115
Synonym: Decapryn
Target: Histamine Receptor
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TargetMol