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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7477 | Antazoline | Others | |
Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias. | |||
T9353 | OXOMEMAZINE | AChR , Histamine Receptor | |
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ... | |||
T36949 | Niaprazine | 5-HT Receptor , Adrenergic Receptor , Histamine Receptor | |
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff... | |||
T1278 | Astemizole | Laridal,Histaminos,Paralergin | Potassium Channel , Histamine Receptor |
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re... | |||
TN1008 | Psoralenoside | CaMK , Calcium Channel , Histamine Receptor | |
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity. | |||
T0147 | Clemastine fumarate | HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate) | Autophagy , Histamine Receptor |
Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties. | |||
T22501 | 2-Pyridylethylamine dihydrochloride | Histamine Receptor | |
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist. | |||
T7085 | Mebhydrolin | Mebhydroline | Histamine Receptor |
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist. | |||
T1469 | Levocetirizine | Levocetirizine HCl | Histamine Receptor |
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist. | |||
T0263 | Chloropyramine hydrochloride | Nilfan,Alergosan,Halopyramine hydrochloride | FAK , VEGFR , Histamine Receptor |
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist. | |||
T23297 | (S)-(+)-Dimethindene maleate | AChR , Histamine Receptor | |
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M4 receptors. | |||
T13566 | Bamirastine | TAK-427 | Histamine Receptor |
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on allergic skin inflammation. | |||
T22842 | HTMT dimaleate | Histamine Trifluoromethyl Toluidide Dimaleate | Histamine Receptor |
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist. | |||
T6426 | Buclizine dihydrochloride | Longifene,Buclina,Buclizine HCl,UCB-4445 | 5-HT Receptor , AChR , Histamine Receptor |
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ... | |||
T1097 | Loratadine | SCH 29851,Loratidine | Influenza Virus , Histamine Receptor |
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical antihistamines (HISTAMINE H1 ANTAGONISTS) it lacks central ne... | |||
T22354 | Levocetirizine Dihydrochloride | Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride | Histamine Receptor |
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro... | |||
T0092 | Antazoline hydrochloride | Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl | Histamine Receptor |
Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous histamine. | |||
T20884 | Hydroxyzine | Hydroxyzine free base | Histamine Receptor |
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor. | |||
T7893 | Bepotastine | Bepotastine free base | Others , Histamine Receptor |
Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis. | |||
T1115 | Doxylamine succinate | Decapryn | Histamine Receptor |
Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties. Doxylamine succinate (Decapryn) competitively blocks the histamine H1 receptor and limits the typical allergic and ... |